Table II.

TZD induced changes in the free energy of dimerization of gA channels

TZD ΔGtot gA-(13)MD SD ΔGtot AgA(15)MD SD 
1 µM troglitazone −5.0 0.60 −4.0 0.8 
30 µM rosiglitazone −5.0 0.2 −4.0 0.9 
10 µM pioglitazone −4.6 1.2 −4.2 1.3 
6 µM ciglitazone 1.7 1.7 −0.6 2.4 
TZD ΔGtot gA-(13)MD SD ΔGtot AgA(15)MD SD 
1 µM troglitazone −5.0 0.60 −4.0 0.8 
30 µM rosiglitazone −5.0 0.2 −4.0 0.9 
10 µM pioglitazone −4.6 1.2 −4.2 1.3 
6 µM ciglitazone 1.7 1.7 −0.6 2.4 

Results in kJ/mole, n = 2–4.

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