TABLE III.
Gating Parameters Based on Limiting Slope logP
0
α
WT
α
D369G
L
0
1.12 ± 0.02e
−6
2.49 ± 0.08e
−6
K
C
(μM)
8.7 ± 0.8
3.8 ± 1.0
K
O
(μM)
1.0 ± 0.2
0.5 ± 0.1
C
8.7 ± 0.8
7.5 ± 0.8
α
WT
α
D369G
L
0
1.12 ± 0.02e
−6
2.49 ± 0.08e
−6
K
C
(μM)
8.7 ± 0.8
3.8 ± 1.0
K
O
(μM)
1.0 ± 0.2
0.5 ± 0.1
C
8.7 ± 0.8
7.5 ± 0.8
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