TABLE IV.

Residue 18 coupling potential analysis

Mutant Tau on, msec Tau recovery, msec ΔG(τon), kT ΔG(τrecov), kT On slope, ΔkT/(+) Recov slope, ΔkT/(+) 
V135K/R18 22.8 ± 1.3 (n = 12)a 134.8 ± 4.4 (n = 12) 3.13 ± 0.06 4.90 ± 0.03   
V135K/R18A 61.8 ± 0.89 (n = 4)a 150.8 ± 2.8 (n = 4)a 4.12 ± 0.01 5.02 ± 0.02 −0.96 −0.22 
V135K/R18E 117.6 ± 8.6 (n = 3)b 168 ± 21 (n = 3) 4.80 ± 0.07 5.12 ± 0.13   
V135/R18 29.5 ± 0.16 (n = 17) 138.8 ± 4.9 (n = 27) 3.38 ± 0.01 4.93 ± 0.04   
V135/R18A 98 ± 3.8 (n = 12)a 123 ± 5.6 (n = 5)b 4.58 ± 0.04 4.81 ± 0.05 −1.28 −0.05 
V135/R18E 401.6 ± 15.7 (n = 16)a 127.4 ± 5.6 (n = 15)a 6.00 ± 0.04 4.85 ± 0.04   
V135D/R18 39.2 ± 1.5 (n = 3)a 166.4 ± 6.5 (n = 3)a 3.67 ± 0.04 5.11 ± 0.04   
V135D/R18A 258 ± 15.2 (n = 10)a 133.3 ± 7 (n = 9)b 5.55 ± 0.06 4.89 ± 0.05 −1.63 −0.20 
V135D/R18E 1006 ± 75 (n = 10)a 116.8 ± 2.7 (n = 10)b 6.91 ± 0.07 4.76 ± 0.02   
KKK/R18 321 ± 9.5 (n = 16)a 286.5 ± 12.4 (n = 13)a 5.77 ± 0.03 5.66 ± 0.04   
KKK/R18A 465.7 ± 15.4 (n = 9)a 328.2 ± 14.2 (n = 4) 6.14 ± 0.03 5.79 ± 0.04 −0.14 0.00 
KKK/R18E 428 ± 16.7 (n = 6)a 289 ± 13 (n = 6) 6.06 ± 0.04 5.67 ± 0.04   
AAA/R18 44.5 ± 0.8 (n = 3)a 152.5 ± 7.4 (n = 3)a 3.80 ± 0.02 5.03 ± 0.05   
AAA/R18A 101.8 ± 4 (n = 6)a 208.1 ± 9.9 (n = 6)a 4.62 ± 0.04 5.33 ± 0.05 −0.53 −0.13 
AAA/R18E 113.9 ± 4 (n = 6)a 203.4 ± 4.5 (n = 6)b 4.74 ± 0.04 5.32 ± 0.02   
EDE/R18 29.5 ± 0.16 (n = 17) 138.8 ± 4.9 (n = 27) 3.38 ± 0.01 4.93 ± 0.04   
EDE/R18A 98 ± 3.8 (n = 12)a 123 ± 5.6 (n = 5)b 4.58 ± 0.04 4.81 ± 0.05 −1.28 −0.05 
EDE/R18E 401.6 ± 15.7 (n = 16)a 127.4 ± 5.6 (n = 15)a 6.00 ± 0.04 4.85 ± 0.04   
Mutant Tau on, msec Tau recovery, msec ΔG(τon), kT ΔG(τrecov), kT On slope, ΔkT/(+) Recov slope, ΔkT/(+) 
V135K/R18 22.8 ± 1.3 (n = 12)a 134.8 ± 4.4 (n = 12) 3.13 ± 0.06 4.90 ± 0.03   
V135K/R18A 61.8 ± 0.89 (n = 4)a 150.8 ± 2.8 (n = 4)a 4.12 ± 0.01 5.02 ± 0.02 −0.96 −0.22 
V135K/R18E 117.6 ± 8.6 (n = 3)b 168 ± 21 (n = 3) 4.80 ± 0.07 5.12 ± 0.13   
V135/R18 29.5 ± 0.16 (n = 17) 138.8 ± 4.9 (n = 27) 3.38 ± 0.01 4.93 ± 0.04   
V135/R18A 98 ± 3.8 (n = 12)a 123 ± 5.6 (n = 5)b 4.58 ± 0.04 4.81 ± 0.05 −1.28 −0.05 
V135/R18E 401.6 ± 15.7 (n = 16)a 127.4 ± 5.6 (n = 15)a 6.00 ± 0.04 4.85 ± 0.04   
V135D/R18 39.2 ± 1.5 (n = 3)a 166.4 ± 6.5 (n = 3)a 3.67 ± 0.04 5.11 ± 0.04   
V135D/R18A 258 ± 15.2 (n = 10)a 133.3 ± 7 (n = 9)b 5.55 ± 0.06 4.89 ± 0.05 −1.63 −0.20 
V135D/R18E 1006 ± 75 (n = 10)a 116.8 ± 2.7 (n = 10)b 6.91 ± 0.07 4.76 ± 0.02   
KKK/R18 321 ± 9.5 (n = 16)a 286.5 ± 12.4 (n = 13)a 5.77 ± 0.03 5.66 ± 0.04   
KKK/R18A 465.7 ± 15.4 (n = 9)a 328.2 ± 14.2 (n = 4) 6.14 ± 0.03 5.79 ± 0.04 −0.14 0.00 
KKK/R18E 428 ± 16.7 (n = 6)a 289 ± 13 (n = 6) 6.06 ± 0.04 5.67 ± 0.04   
AAA/R18 44.5 ± 0.8 (n = 3)a 152.5 ± 7.4 (n = 3)a 3.80 ± 0.02 5.03 ± 0.05   
AAA/R18A 101.8 ± 4 (n = 6)a 208.1 ± 9.9 (n = 6)a 4.62 ± 0.04 5.33 ± 0.05 −0.53 −0.13 
AAA/R18E 113.9 ± 4 (n = 6)a 203.4 ± 4.5 (n = 6)b 4.74 ± 0.04 5.32 ± 0.02   
EDE/R18 29.5 ± 0.16 (n = 17) 138.8 ± 4.9 (n = 27) 3.38 ± 0.01 4.93 ± 0.04   
EDE/R18A 98 ± 3.8 (n = 12)a 123 ± 5.6 (n = 5)b 4.58 ± 0.04 4.81 ± 0.05 −1.28 −0.05 
EDE/R18E 401.6 ± 15.7 (n = 16)a 127.4 ± 5.6 (n = 15)a 6.00 ± 0.04 4.85 ± 0.04   

aP < 0.01 and bP < 0.05. R18 mutants compared to V135K or EDE(161-3)KKK parent constructs, respectively; R18 plus EDE(161-3)KKK or V135K constructs compared to wild type.

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