TABLE I

BKCa Channel Ca2+ Binding Parameters

Binding Site
Membrane Potential (mV)
KC (μM)
KO (μM)
M
f
C
Ca2+ Bowl       
    ΔEΔR −80 3.1 ± 0.2 0.88 ± 0.06   3.55 
    ΔEΔR 3.1 0.88   3.55 
RCK1       
    ΔEΔB(D2A2) −80 23.2 ± 2.6 4.9 ± 0.6   4.75 
    ΔEΔB(D5N5) −80 26.8 ± 3.8 5.6 ± 0.8   4.75 
    ΔEΔB(D2A2) + Cooperativity −80 13.7 ± 2.3 2.8 ± 0.5  0.45 ± 0.1  
    ΔEΔB(D5N5)+ Cooperativity −80 9.4 ± 1.8 1.8 ± 0.2  0.27 ± 0.05  
    ΔEΔB(D2A2) 15.8 ± 3.1 2.10 ± 0.4 1.8 × 107  7.52  
Binding Site
Membrane Potential (mV)
KC (μM)
KO (μM)
M
f
C
Ca2+ Bowl       
    ΔEΔR −80 3.1 ± 0.2 0.88 ± 0.06   3.55 
    ΔEΔR 3.1 0.88   3.55 
RCK1       
    ΔEΔB(D2A2) −80 23.2 ± 2.6 4.9 ± 0.6   4.75 
    ΔEΔB(D5N5) −80 26.8 ± 3.8 5.6 ± 0.8   4.75 
    ΔEΔB(D2A2) + Cooperativity −80 13.7 ± 2.3 2.8 ± 0.5  0.45 ± 0.1  
    ΔEΔB(D5N5)+ Cooperativity −80 9.4 ± 1.8 1.8 ± 0.2  0.27 ± 0.05  
    ΔEΔB(D2A2) 15.8 ± 3.1 2.10 ± 0.4 1.8 × 107  7.52  

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