Table I.

Binding characteristics of Evasin-1 and -3 as determined by SPR

CKBP
Chemokine
ka × 106
kd × 10−3
Kd × 10−9


M−1s−1
s−1
nM
Evasin-1 CCL3 13.8 ± 3.54 2.43 ± 0.61 0.12 
 CCL3L1 13.2 ± 2.9 0.67 ± 0.13 0.05 
 mMIP-1α 15.6 ± 16 1.18 ± 1.07 0.08 
 CCL4 4.29 ± 2.58 2.2 ± 0.18 0.51 
 mMIP-1β 3.84 ± 1.42 0.58 ± 0.12 0.15 
Evasin-3 (HEK) CXCL1 3.95 ± 4.23 1.42 ± 0.36 0.34 
 CXCL8 0.41 ± 0.30 0.29 ± 0.14 0.7 
 KC 0.64 ± 0.58 1.44 ± 0.35 2.25 
 MIP-2 0.79 ± 0.9 0.33 ± 0.11 0.4 
Evasin-3 (E. coliCXCL1 2.61 ± 0.69 2.22 ± 0.49 0.85 
 CXCL8 0.84 ± 0.33 0.36 ± 0.05 0.43 
 KC 0.32 ± 0.17 1.85 ± 0.43 5.78 
 MIP-2 1.02 ± 0.56 0.65 ± 0.25 0.64 
CKBP
Chemokine
ka × 106
kd × 10−3
Kd × 10−9


M−1s−1
s−1
nM
Evasin-1 CCL3 13.8 ± 3.54 2.43 ± 0.61 0.12 
 CCL3L1 13.2 ± 2.9 0.67 ± 0.13 0.05 
 mMIP-1α 15.6 ± 16 1.18 ± 1.07 0.08 
 CCL4 4.29 ± 2.58 2.2 ± 0.18 0.51 
 mMIP-1β 3.84 ± 1.42 0.58 ± 0.12 0.15 
Evasin-3 (HEK) CXCL1 3.95 ± 4.23 1.42 ± 0.36 0.34 
 CXCL8 0.41 ± 0.30 0.29 ± 0.14 0.7 
 KC 0.64 ± 0.58 1.44 ± 0.35 2.25 
 MIP-2 0.79 ± 0.9 0.33 ± 0.11 0.4 
Evasin-3 (E. coliCXCL1 2.61 ± 0.69 2.22 ± 0.49 0.85 
 CXCL8 0.84 ± 0.33 0.36 ± 0.05 0.43 
 KC 0.32 ± 0.17 1.85 ± 0.43 5.78 
 MIP-2 1.02 ± 0.56 0.65 ± 0.25 0.64 

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