| Construct | EC50 (µM) | Slope, n | IC50 (mM) | Slope, b | Cells (no.) |
|---|---|---|---|---|---|
| K2(Q) WT (KA-evoked) | 0.89 ± 0.08 | 1.1 ± 0.1 | 5 | ||
| K2(R) WT (KA-evoked) | 0.25 ± 0.04 | 1.0 ± 0.1 | 4 | ||
| K2(Q&R) A8C | 7.3 ± 1.4 | 1.6 ± 0.4 | 25 ± 5.4 | 1.3 ± 0.4 | 23 |
| K2(Q) L10C | 1,800 ± 300 | 1.2 ± 0.2 | 26 ± 7.1 | 1.9 ± 0.5 | 12 |
| N1/K2 A8C + N2B/K2 A8C | 5.6 ± 1.7 | 0.9 ± 0.1 | 1.1 ± 0.2 | 1.8 ± 0.4 | 21 |
| N1/K2 A8C + N2B/K2 | 47 ± 8 | 1.0 ± 0.2 | 13 ± 10 | 0.9 ± 0.4 | 14 |
| N1/K2 + N2B/K2 A8C | 27 ± 9 | 0.9 ± 0.1 | 1.1 ± 0.2 | 1.8 ± 0.4 | 14 |
| K2(Q) WT (KA-evoked) | 0.89 ± 0.08 | 1.1 ± 0.1 | 5 | ||
| K2(R) WT (KA-evoked) | 0.25 ± 0.04 | 1.0 ± 0.1 | 4 | ||
| K2(Q&R) A8C | 7.3 ± 1.4 | 1.6 ± 0.4 | 25 ± 5.4 | 1.3 ± 0.4 | 23 |
| K2(Q) L10C | 1,800 ± 300 | 1.2 ± 0.2 | 26 ± 7.1 | 1.9 ± 0.5 | 12 |
| N1/K2 A8C + N2B/K2 A8C | 5.6 ± 1.7 | 0.9 ± 0.1 | 1.1 ± 0.2 | 1.8 ± 0.4 | 21 |
| N1/K2 A8C + N2B/K2 | 47 ± 8 | 1.0 ± 0.2 | 13 ± 10 | 0.9 ± 0.4 | 14 |
| N1/K2 + N2B/K2 A8C | 27 ± 9 | 0.9 ± 0.1 | 1.1 ± 0.2 | 1.8 ± 0.4 | 14 |
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