Table 2.
Pyramid skew and agonist orientation,
A
R* versus
A
R homology structures (α−γ)
Agonist
.
ΔΘ
s
(degrees)
.
Θ
a
R*
(degrees)
.
Θ
a
R
(degrees)
.
ACh
2.9
292.7 ± 9.8
125.2 ± 8.9
CCh
2.8
288.3 ± 9.3
123.9 ± 6.4
TMA
2.7
-
-
Cho
2.7
104.5 ± 7.6
126.4 ± 6.5
Agonist
.
ΔΘ
s
(degrees)
.
Θ
a
R*
(degrees)
.
Θ
a
R
(degrees)
.
ACh
2.9
292.7 ± 9.8
125.2 ± 8.9
CCh
2.8
288.3 ± 9.3
123.9 ± 6.4
TMA
2.7
-
-
Cho
2.7
104.5 ± 7.6
126.4 ± 6.5
Positive ΔΘ
s
is counterclockwise.
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