Table 4.
Spermine block rates in GluA2 receptors with auxiliary proteins
ReceptorTwo-conductance permeant blocker modeln
konkoffkpermk1k1'Kd(0mV)
a (µM−1s−1)b (mV)c (s−1)d (mV)e (s−1)f (mV)(µM)
GluA2 31 199  184 -20  23 19  4.55E+09 2.95E+07 3.3 
SEM 94  44   1.93E+09 2.04E+07 0.5  
GluA2-γ2 24 369  499 -13  131 16  1.67E+08 4.16E+07 15 
SEM 223  147  25  1.64E+08 4.12E+07  
GluA2 + CNIH-3 44 291  313 -19  53 15  2.10E+09 1.29E+06 4.5 
SEM 16 139  81  29  1.98E+09 1.06E+06 0.9  
ReceptorTwo-conductance permeant blocker modeln
konkoffkpermk1k1'Kd(0mV)
a (µM−1s−1)b (mV)c (s−1)d (mV)e (s−1)f (mV)(µM)
GluA2 31 199  184 -20  23 19  4.55E+09 2.95E+07 3.3 
SEM 94  44   1.93E+09 2.04E+07 0.5  
GluA2-γ2 24 369  499 -13  131 16  1.67E+08 4.16E+07 15 
SEM 223  147  25  1.64E+08 4.12E+07  
GluA2 + CNIH-3 44 291  313 -19  53 15  2.10E+09 1.29E+06 4.5 
SEM 16 139  81  29  1.98E+09 1.06E+06 0.9  

Block rate parameters were obtained by fitting the current relaxation after the voltage steps.

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