Table 3.
Spermine block rates in GluA2 receptors
ReceptorPermeant blocker modeln
konkoffkpermKd(0mV)
a (µM−1s−1)b (mV)c (s−1)d (mV)e (s−1)f (mV)(µM)
GluA2 29 113  156 −19  32 20  
SEM 13  30  16   
ReceptorPermeant blocker modeln
konkoffkpermKd(0mV)
a (µM−1s−1)b (mV)c (s−1)d (mV)e (s−1)f (mV)(µM)
GluA2 29 113  156 −19  32 20  
SEM 13  30  16   

Block rate parameters were obtained by fitting the current relaxation after the voltage steps.

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