Table 1.

Mean ± SEM for parameters used to fit ADP concentration-response relationships for the indicated KATP channels in the presence or absence of sulfonylureas

Channel Parameter Mg2+ No sulfonylurea +Sulfonylurea 
30 µM gliclazide     
Kir6.2/SUR1 IC50 (µM) − 62 ± 3 (n = 6) 59 ± 7 (n = 6) 
Kir6.2/SUR1 IC50 (µM) 258 ± 57 (n = 12) 64 ± 3a (n = 6) 
Kir6.2/SUR1 EC50 (µM) 13 ± 2 (n = 12) n.a. 
Kir6.2/SUR1 a 3.2 ± 0.7 (n = 12) n.a. 
Kir.2/SUR2A-YS IC50 (µM) − 95 ± 5 (n = 6) 88 ± 11 (n = 6) 
Kir.2/SUR2A-YS IC50 (µM) 310 ± 56 (n = 6) 286 ± 39 (n = 6) 
Kir.2/SUR2A-YS EC50 (µM) 16 ± 5 (n = 6) 19 ± 3 (n = 6) 
Kir.2/SUR2A-YS a 1.2 ± 0.3 (n = 6) 1.1 ± 0.1 (n = 6) 
1 µM glibenclamide     
Kir6.2/SUR2A IC50 (µM) − 96 ± 19 (n = 6) 80 ± 8 (n = 6) 
Kir6.2/SUR2A IC50 (µM) 280 ± 70 (n = 7) 315 ± 49 (n = 7) 
Kir6.2/SUR2A EC50 (µM) 22 ± 8 (n = 7) 17 ± 2 (n = 7) 
Kir6.2/SUR2A a 1.1 ± 0.3 (n = 7) 1.1 ± 0.2 (n = 7) 
Channel Parameter Mg2+ No sulfonylurea +Sulfonylurea 
30 µM gliclazide     
Kir6.2/SUR1 IC50 (µM) − 62 ± 3 (n = 6) 59 ± 7 (n = 6) 
Kir6.2/SUR1 IC50 (µM) 258 ± 57 (n = 12) 64 ± 3a (n = 6) 
Kir6.2/SUR1 EC50 (µM) 13 ± 2 (n = 12) n.a. 
Kir6.2/SUR1 a 3.2 ± 0.7 (n = 12) n.a. 
Kir.2/SUR2A-YS IC50 (µM) − 95 ± 5 (n = 6) 88 ± 11 (n = 6) 
Kir.2/SUR2A-YS IC50 (µM) 310 ± 56 (n = 6) 286 ± 39 (n = 6) 
Kir.2/SUR2A-YS EC50 (µM) 16 ± 5 (n = 6) 19 ± 3 (n = 6) 
Kir.2/SUR2A-YS a 1.2 ± 0.3 (n = 6) 1.1 ± 0.1 (n = 6) 
1 µM glibenclamide     
Kir6.2/SUR2A IC50 (µM) − 96 ± 19 (n = 6) 80 ± 8 (n = 6) 
Kir6.2/SUR2A IC50 (µM) 280 ± 70 (n = 7) 315 ± 49 (n = 7) 
Kir6.2/SUR2A EC50 (µM) 22 ± 8 (n = 7) 17 ± 2 (n = 7) 
Kir6.2/SUR2A a 1.1 ± 0.3 (n = 7) 1.1 ± 0.2 (n = 7) 

Parameters were obtained from the data shown in Fig. 4, but all values are the mean of the fits to the individual dose–response curves. a is the maximal increase in KATP current caused by MgADP activation (Eq. 4; note the maximal amplitude of activation is given by 1 + a). n.a., not applicable.

a

P < 0.01 against control (Student’s t test).

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