Table 1.

Equations for minimal PI(4,5)P2–DAG reaction scheme

Equation No. 
d[PI(4,5)P2]local=d[PI(4,5)P2]locald[PI(4,5)P2]local·ki(t)·Def(t)·dt 
d[DAG]=d[DAG]+d[PI(4,5)P2]tot·ki(t)·Def(t)·dtd[DAG]·kii·dt 
d[IP3]=d[IP3]+d[PI(4,5)P2]tot·ki(t)·Def(t)·dtd[IP3]·kv·dt 
Def(t)=1(Rd_f·exp(τrd)/t)+Sd_f·exp(τsd/t)Rd_f:fraction of rapid desensitizationSd_f:fraction of slow desensitizationτrd:time constant for the rapid desensitizationτsd:time constant for the slow desensitization 
ki(t)=ki·B_PLCpgtB_PLC:basal PLC activitypg:power parameter ofGqPCR receptor stimulation 10 
d[PA]=d[PA]+d[DAG]·kii·dtd[PA]·kiii·dt 11 
d[PI(4)P]=d[PI(4)P]+d[PA]·kiii·dtd[PI(4)P]·kiv·dt 12 
d[PI(4,5)P2]recovered=d[PI(4)P]·kiv·dtd[PI(4,5)P2]recovered·ki(t)·Def(t)·dt 13 
d[PI(4,5)P2]global=d[PI(4,5)P2]globald[PI(4,5)P2]global·ki_g(t)·Def(t)·dtki_g:rate constant for global PLC activity 14 
d[PI(4,5)P2]diffused_in=(d[PI(4,5)P2]globald[PI(4,5)P2]local)·(1errf(spot/sprt(4·dcoef·dt)))d[PI(4,5)P2]diffused_in·ki(t)· Def(t)· dterrf:error functiondcoef:diffusion coefficient of PI(4,5)P2spot:distance between local and global domain 15 
d[PI(4,5)P2]scavenged_PHd=(d[PHd]reld[PHd]IP3)·(1/(1+Kd,PHd/(d[PI(4,5)P2]local+d[PI(4,5)P2]recovered+d[PI(4,5)P2]diffused_in))) 16 
d[PI(4,5)P2]tot=d[PI(4,5)P2]local+d[PI(4,5)P2]recovered+d[PI(4,5)P2]diffused_ind[PI(4,5)P2]scavenged_PHd 17 
Equation No. 
d[PI(4,5)P2]local=d[PI(4,5)P2]locald[PI(4,5)P2]local·ki(t)·Def(t)·dt 
d[DAG]=d[DAG]+d[PI(4,5)P2]tot·ki(t)·Def(t)·dtd[DAG]·kii·dt 
d[IP3]=d[IP3]+d[PI(4,5)P2]tot·ki(t)·Def(t)·dtd[IP3]·kv·dt 
Def(t)=1(Rd_f·exp(τrd)/t)+Sd_f·exp(τsd/t)Rd_f:fraction of rapid desensitizationSd_f:fraction of slow desensitizationτrd:time constant for the rapid desensitizationτsd:time constant for the slow desensitization 
ki(t)=ki·B_PLCpgtB_PLC:basal PLC activitypg:power parameter ofGqPCR receptor stimulation 10 
d[PA]=d[PA]+d[DAG]·kii·dtd[PA]·kiii·dt 11 
d[PI(4)P]=d[PI(4)P]+d[PA]·kiii·dtd[PI(4)P]·kiv·dt 12 
d[PI(4,5)P2]recovered=d[PI(4)P]·kiv·dtd[PI(4,5)P2]recovered·ki(t)·Def(t)·dt 13 
d[PI(4,5)P2]global=d[PI(4,5)P2]globald[PI(4,5)P2]global·ki_g(t)·Def(t)·dtki_g:rate constant for global PLC activity 14 
d[PI(4,5)P2]diffused_in=(d[PI(4,5)P2]globald[PI(4,5)P2]local)·(1errf(spot/sprt(4·dcoef·dt)))d[PI(4,5)P2]diffused_in·ki(t)· Def(t)· dterrf:error functiondcoef:diffusion coefficient of PI(4,5)P2spot:distance between local and global domain 15 
d[PI(4,5)P2]scavenged_PHd=(d[PHd]reld[PHd]IP3)·(1/(1+Kd,PHd/(d[PI(4,5)P2]local+d[PI(4,5)P2]recovered+d[PI(4,5)P2]diffused_in))) 16 
d[PI(4,5)P2]tot=d[PI(4,5)P2]local+d[PI(4,5)P2]recovered+d[PI(4,5)P2]diffused_ind[PI(4,5)P2]scavenged_PHd 17 

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