Table 1.

Voltage-dependent activation of HCN channels

Cell type, channel, recording configuration Activation midpoint ΔV1/2 
 Control cAMP  
 mV mV mV 
CHO, HCN4, whole cell −106.3 ± 2.7 (9) −106.6 ± 3.8 (7)a −0.3 
CHO, HCN2, whole cell −107.7 ± 3.4 (9) −91.8 ± 2.7 (10)b +15.9 
HEK, HCN4, whole cell −121.6 ± 5.3 (8)c −104.3 ± 1.6 (7)b +17.3 
HEK, HCN4-R669Q, whole cell −123.5 ± 1.2 (7) −120.1 ± 2.3 (11)a +3.4 
CHO, HCN4, patches −120.2 ± 3.7 (8) −118.7 ± 2.8 (8)a +1.5 ± 1.8 (8) 
HEK, HCN4, patches −137.2 ± 2.2 (6)c −126.1 ± 2.8 (6)b + 11.1 ± 1.0 (6) 
CHO, HCN2, patches −118.2 ± 2.9 (5) −101.1 ± 2.7 (5)b +17.1 ± 0.4 (5) 
CHO, HCN4-2Tail, whole cell −118.9 ± 2.5 (4) −105.4 ± 3.0 (5)b +13.5 
CHO, HCN2-4Tail, whole cell −110.2 ± 2.9 (6) −78.9 ± 4.3 (4)b +31.3 
CHO, HCN4-Δ719, whole cell −122.9 ± 2.2 (7)c −106.7 ± 2.9 (8)b +16.2 
CHO, HCN4-Δ1012, whole cell −109.2 ± 1.5 (7) −106.0 ± 1.5 (7)a +3.2 
Cell type, channel, recording configuration Activation midpoint ΔV1/2 
 Control cAMP  
 mV mV mV 
CHO, HCN4, whole cell −106.3 ± 2.7 (9) −106.6 ± 3.8 (7)a −0.3 
CHO, HCN2, whole cell −107.7 ± 3.4 (9) −91.8 ± 2.7 (10)b +15.9 
HEK, HCN4, whole cell −121.6 ± 5.3 (8)c −104.3 ± 1.6 (7)b +17.3 
HEK, HCN4-R669Q, whole cell −123.5 ± 1.2 (7) −120.1 ± 2.3 (11)a +3.4 
CHO, HCN4, patches −120.2 ± 3.7 (8) −118.7 ± 2.8 (8)a +1.5 ± 1.8 (8) 
HEK, HCN4, patches −137.2 ± 2.2 (6)c −126.1 ± 2.8 (6)b + 11.1 ± 1.0 (6) 
CHO, HCN2, patches −118.2 ± 2.9 (5) −101.1 ± 2.7 (5)b +17.1 ± 0.4 (5) 
CHO, HCN4-2Tail, whole cell −118.9 ± 2.5 (4) −105.4 ± 3.0 (5)b +13.5 
CHO, HCN2-4Tail, whole cell −110.2 ± 2.9 (6) −78.9 ± 4.3 (4)b +31.3 
CHO, HCN4-Δ719, whole cell −122.9 ± 2.2 (7)c −106.7 ± 2.9 (8)b +16.2 
CHO, HCN4-Δ1012, whole cell −109.2 ± 1.5 (7) −106.0 ± 1.5 (7)a +3.2 
a

Not significantly different (P > 0.05) compared to corresponding control.

b

Significantly different (P < 0.05) compared to corresponding control.

c

Significantly different (P < 0.05) compared to CHO-HCN4 control in same recording configuration.

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