Table 1.

Shifts in Vmedian and in V1/2 occurring with Cd2+

Parameter Vmedian V1/2 
462C466C QON (0 mM Cd2+−117.9 ± 4.5 −132.7 ± 5.7 
QON (130 mM Cd2+−89.9 ± 10.3 −103.9 ± 8.9 
QOFF (0 mM Cd2+−112.9 ± 3.2 −126.7 ± 4.2 
QOFF (130 mM Cd2+−101.5 ± 4.4 −99.9 ± 5.4 
462Y468C QON (0 mM Cd2+−91.9 ± 8.4 −116.4 ± 4.8 
QON (130 mM Cd2+−104.8 ± 7.9 −131.8 ± 3.9 
QOFF (0 mM Cd2+−94.7 ± 6.5 −96.7 ± 4.6 
QOFF (130 mM Cd2+−106.6 ± 6.4 −128.0 ± 4.2 
Parameter Vmedian V1/2 
462C466C QON (0 mM Cd2+−117.9 ± 4.5 −132.7 ± 5.7 
QON (130 mM Cd2+−89.9 ± 10.3 −103.9 ± 8.9 
QOFF (0 mM Cd2+−112.9 ± 3.2 −126.7 ± 4.2 
QOFF (130 mM Cd2+−101.5 ± 4.4 −99.9 ± 5.4 
462Y468C QON (0 mM Cd2+−91.9 ± 8.4 −116.4 ± 4.8 
QON (130 mM Cd2+−104.8 ± 7.9 −131.8 ± 3.9 
QOFF (0 mM Cd2+−94.7 ± 6.5 −96.7 ± 4.6 
QOFF (130 mM Cd2+−106.6 ± 6.4 −128.0 ± 4.2 

The trapezoid method (Chowdhury and Chanda, 2012) was used to calculate the Vmedian values from locked-open and locked-closed mutants, and V1/2 values were calculated from a single Boltzmann fit.

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