Table 2. Equilibrium constants for wt... | Rockefeller University Press

Table 2.

Equilibrium constants for wt AChRs

Agonists	K_d	J_d	E₂
	M	M
Cho^a	4.1 E-3	15.1 E-6	0.046
DMP	2.1 E-3	2.77 E-6	0.38
DMT	1.6 E-3	1.77 E-6	0.58
Nic	1 E-3	0.95 E-6	0.87
TMA	0.81 E-3	0.41 E-6	2.54
CCh	0.41 E-3	0.14 E-6	5.33
ACh	0.16 E-3	2.65 E-8	25.4

Agonists	K_d	J_d	E₂
	M	M
Cho^a	4.1 E-3	15.1 E-6	0.046
DMP	2.1 E-3	2.77 E-6	0.38
DMT	1.6 E-3	1.77 E-6	0.58
Nic	1 E-3	0.95 E-6	0.87
TMA	0.81 E-3	0.41 E-6	2.54
CCh	0.41 E-3	0.14 E-6	5.33
ACh	0.16 E-3	2.65 E-8	25.4

See Table 1. E₂, the diliganded gating equilibrium constant.

Purohit and Grosman, 2006.