Table 1.
SGC chemical probes: Links to selectivity, cell-based assay, and crystal structure information
DrugTargetSGC link
UNC1999 EZH1 and 2 https://www.thesgc.org/chemical-probes/UNC1999 
JQ1 BRD2, 3, 4 and T https://www.thesgc.org/chemical-probes/JQ1 
A-366 G9a and GLP https://www.thesgc.org/chemical-probes/A-366 
GSKLSD1 LSD1 https://www.thesgc.org/chemical-probes/GSK-LSD1 
PFI-2 SETD7 https://www.thesgc.org/chemical-probes/PFI-2 
PFI-3 SMARCA2, 4 and PB1 https://www.thesgc.org/chemical-probes/PFI-3 
OICR-9429 WDR5 https://www.thesgc.org/chemical-probes/OICR-9429 
GSK2801 BAZ2A and 2B https://www.thesgc.org/chemical-probes/GSK2801 
A-196 SUV420H1 and H2 https://www.thesgc.org/chemical-probes/A-196 
BAY598 SMYD2 https://www.thesgc.org/chemical-probes/BAY-598 
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