Table I.

Values of binding and dissociation rate constants

Value  XPC  TFIIH  XPG  XPA  XPF/ ERCC1  RPA  PCNA  
Concentration (µM)  0.140  0.360  0.440  1.110  0.170  1.110  1.110  
Damaged DNA  
kon (µM−1s−1)  0.008 (0.007; 0.011)  1.6 (0.8; 4.5)  NA  NA  NA  NA  NA  
koff (s−1)  0.061 (0.007; 0.462)  0.053 (0.004; 0.195)  NA  NA  NA  NA  NA  
Kd (µM)  7.8  0.03  NA  NA  NA  NA  NA  
Partially unwound DNA  
kon (µM−1s−1)  0.002 (0.001; 0.003)  0.26 (0.11; 0.27)  0.28 (0.19; 0.31)  0.13 (0.12; 0.16)  1.2 (1.1; 1.6)  0.15 (0.11; 0.22)  NA  
koff (s−1)  0.007 (0.006; 0.008)  0.012 (0.009; 0.016)  0.015 (0.012; 0.015)  1.04 (0.75; 1.30)  0.01 (0.011; 0.014)  2.6 (1.7; 3.6)  NA  
Kd (µM)  3.1  0.05  0.05  7.7  0.01  17  NA  
τ = 35 ± 30 min  
Fully unwound DNA  
kon (µM−1s−1)  0.002 (0.001; 0.003)  0.26 (0.11; 0.27)  0.28 (0.19; 0.31)  0.13 (0.12; 0.16)  1.2 (1.1; 1.6)  0.006 (0.006; 0.007)  NA  
koff (s−1)  0.007 (0.006; 0.008)  0.012 (0.009; 0.016)  0.015 (0.012; 0.015)  1.04 (0.75; 1.30)  0.01 (0.011; 0.014)  0.021 (0.020; 0.022)  NA  
Kd (µM)  3.1  0.05  0.05  7.7  0.01  3.27  NA  
τ = 41 ± 36 min  
Incised DNA  
kon (µM−1s−1)  0.22 (0.13; 0.26)  0.0004 (0.0003; 0.010)  0.001 (0.0004; 0.007)  0.004 (0.004; 0.005)  0.09 (0.07; 0.11)  0.006 (0.006; 0.007)  0.001 (0.001; 0.002)  
koff (s−1)  0.40 (0.21; 0.48)  0.05 (0.04; 0.07)  0.10 (0.04; 0.11)  0.06 (0.05; 0.07)  0.050 (0.040; 0.101)  0.021 (0.020; 0.022)  0.004 (0.004; 0.004)  
Kd (µM)  1.8  137  89  13  0.53  3.27  2.8  
τ = 41 ± 36 min  
Resynthesized DNA  
kon (µM−1s−1)  NA  NA  NA  0.054 (0.054; 0.058)  NA  0.08 (0.05; 0.10)  0.010 (0.007; 0.010)  
koff (s−1)  NA  NA  NA  0.004 (0.004; 0.005)  NA  0.04 (0.03; 0.05)  0.002 (0.002; 0.002)  
Kd (µM)  NA  NA  NA  0.08  NA  0.51  0.19  
τ = 2.0 ± 0.7 h  
Rechromatinized DNA  
kon (µM−1s−1)  NA  NA  NA  NA  NA  0.07 (0.06; 0.07)  0.31 (0.25; 0.34)  
koff (s−1)  NA  NA  NA  NA  NA  0.04 (0.04; 0.05)  0.05 (0.04; 0.05)  
Kd (µM)  NA  NA  NA  NA  NA  0.61  0.16  
τ = 2.2 ± 0.7 h  
Value  XPC  TFIIH  XPG  XPA  XPF/ ERCC1  RPA  PCNA  
Concentration (µM)  0.140  0.360  0.440  1.110  0.170  1.110  1.110  
Damaged DNA  
kon (µM−1s−1)  0.008 (0.007; 0.011)  1.6 (0.8; 4.5)  NA  NA  NA  NA  NA  
koff (s−1)  0.061 (0.007; 0.462)  0.053 (0.004; 0.195)  NA  NA  NA  NA  NA  
Kd (µM)  7.8  0.03  NA  NA  NA  NA  NA  
Partially unwound DNA  
kon (µM−1s−1)  0.002 (0.001; 0.003)  0.26 (0.11; 0.27)  0.28 (0.19; 0.31)  0.13 (0.12; 0.16)  1.2 (1.1; 1.6)  0.15 (0.11; 0.22)  NA  
koff (s−1)  0.007 (0.006; 0.008)  0.012 (0.009; 0.016)  0.015 (0.012; 0.015)  1.04 (0.75; 1.30)  0.01 (0.011; 0.014)  2.6 (1.7; 3.6)  NA  
Kd (µM)  3.1  0.05  0.05  7.7  0.01  17  NA  
τ = 35 ± 30 min  
Fully unwound DNA  
kon (µM−1s−1)  0.002 (0.001; 0.003)  0.26 (0.11; 0.27)  0.28 (0.19; 0.31)  0.13 (0.12; 0.16)  1.2 (1.1; 1.6)  0.006 (0.006; 0.007)  NA  
koff (s−1)  0.007 (0.006; 0.008)  0.012 (0.009; 0.016)  0.015 (0.012; 0.015)  1.04 (0.75; 1.30)  0.01 (0.011; 0.014)  0.021 (0.020; 0.022)  NA  
Kd (µM)  3.1  0.05  0.05  7.7  0.01  3.27  NA  
τ = 41 ± 36 min  
Incised DNA  
kon (µM−1s−1)  0.22 (0.13; 0.26)  0.0004 (0.0003; 0.010)  0.001 (0.0004; 0.007)  0.004 (0.004; 0.005)  0.09 (0.07; 0.11)  0.006 (0.006; 0.007)  0.001 (0.001; 0.002)  
koff (s−1)  0.40 (0.21; 0.48)  0.05 (0.04; 0.07)  0.10 (0.04; 0.11)  0.06 (0.05; 0.07)  0.050 (0.040; 0.101)  0.021 (0.020; 0.022)  0.004 (0.004; 0.004)  
Kd (µM)  1.8  137  89  13  0.53  3.27  2.8  
τ = 41 ± 36 min  
Resynthesized DNA  
kon (µM−1s−1)  NA  NA  NA  0.054 (0.054; 0.058)  NA  0.08 (0.05; 0.10)  0.010 (0.007; 0.010)  
koff (s−1)  NA  NA  NA  0.004 (0.004; 0.005)  NA  0.04 (0.03; 0.05)  0.002 (0.002; 0.002)  
Kd (µM)  NA  NA  NA  0.08  NA  0.51  0.19  
τ = 2.0 ± 0.7 h  
Rechromatinized DNA  
kon (µM−1s−1)  NA  NA  NA  NA  NA  0.07 (0.06; 0.07)  0.31 (0.25; 0.34)  
koff (s−1)  NA  NA  NA  NA  NA  0.04 (0.04; 0.05)  0.05 (0.04; 0.05)  
Kd (µM)  NA  NA  NA  NA  NA  0.61  0.16  
τ = 2.2 ± 0.7 h  

NA, not applicable. The values for the different repair proteins are arranged in columns for the different DNA repair intermediates to which they bind (rows). The dissociation constants Kd = koff/kon are also given. Reference parameter set and 90% confidence intervals (in parentheses) are shown. Nuclear concentration (in micromolars) of NER factors XPC, XPA, and XPG are based on previously described data (Araújo et al., 2001), whereas RPA and PCNA amounts are estimated to be 250,000 molecules per cell, and TFIIH and ERCC1-XPF were estimated at 65,000 and 50,000 molecules per cell, respectively, based on previous estimates (Houtsmuller et al., 1999; Moné et al., 2004). Concentrations are calculated assuming a nuclear volume of 0.3 pL.

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