Table 2.

The functional effects of Shaker and Kv1.2 mutations

ShakerFunctional effectKv1.2Functional effect
WT W434 Conducting W366 Conducting 
p2 W434F Non-conducting W366F Faster inactivation 
p3 W435F Conducting W367F Conducting 
p4 T439V Non-conducting S371V Faster inactivation 
p5 Y445F
Y445A 
Faster inactivation
Non-conducting 
Y377F
Y377A 
Conducting
Non-conducting 
p6 D447N Non-conducting D379N Non-functional channel 
p7 T449V
T449A
T449K 
Slower inactivation
Faster inactivation
Faster inactivation 
V381T
V381A
V381K 
Conducting
Faster inactivation
Faster inactivation 
p1/p7   Q357A/V381T Conducting 
p2/p7 W434F/T449 Faster inactivation W366F/V381T Non-conducting 
p4/p5   S371T/Y377F Conducting 
p4/p5/p7   S371T/Y377F/V381T Faster inactivation 
p4/p7   S371V/V381T
S371T/V381T 
Non-conducting
Conducting 
p5/p7   Y377F/V381T Faster inactivation 
ShakerFunctional effectKv1.2Functional effect
WT W434 Conducting W366 Conducting 
p2 W434F Non-conducting W366F Faster inactivation 
p3 W435F Conducting W367F Conducting 
p4 T439V Non-conducting S371V Faster inactivation 
p5 Y445F
Y445A 
Faster inactivation
Non-conducting 
Y377F
Y377A 
Conducting
Non-conducting 
p6 D447N Non-conducting D379N Non-functional channel 
p7 T449V
T449A
T449K 
Slower inactivation
Faster inactivation
Faster inactivation 
V381T
V381A
V381K 
Conducting
Faster inactivation
Faster inactivation 
p1/p7   Q357A/V381T Conducting 
p2/p7 W434F/T449 Faster inactivation W366F/V381T Non-conducting 
p4/p5   S371T/Y377F Conducting 
p4/p5/p7   S371T/Y377F/V381T Faster inactivation 
p4/p7   S371V/V381T
S371T/V381T 
Non-conducting
Conducting 
p5/p7   Y377F/V381T Faster inactivation 

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